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Publication Venue For
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Rotational Symmetry of Two Pyrethroid Receptor Sites in the Mosquito Sodium Channel..
88:273-280.
2015
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A mutation in the intracellular loop III/IV of mosquito sodium channel synergizes the effect of mutations in helix IIS6 on pyrethroid resistance..
87:421-429.
2015
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Pro32Pro33 mutations in the integrin β3 PSI domain result in αIIbβ3 priming and enhanced adhesion: reversal of the hypercoagulability phenotype by the Src inhibitor SKI-606..
85:921-931.
2014
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Batrachotoxin, pyrethroids, and BTG 502 share overlapping binding sites on insect sodium channels..
80:426-433.
2011
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The relative activity of "function sparing" HIV-1 entry inhibitors on viral entry and CCR5 internalization: is allosteric functional selectivity a valuable therapeutic property?.
75:490-501.
2009
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Erratum: The NR1 M3 domain mediates allosteric coupling in the N-methyl-D-aspartate receptor (Molecular Pharmacology (2008) 74 (454-465)).
75:255-257.
2009
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N-(6-chloro-pyridin-3-yl)-3,4-difluoro-benzamide (ICA-27243): a novel, selective KCNQ2/Q3 potassium channel activator..
73:977-986.
2008
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Substrate specificities of g protein-coupled receptor kinase-2 and -3 at cardiac myocyte receptors provide basis for distinct roles in regulation of myocardial function..
72:582-591.
2007
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S-nitrosylating agents: a novel class of compounds that increase cystic fibrosis transmembrane conductance regulator expression and maturation in epithelial cells..
70:1435-1442.
2006
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The regulator of G protein signaling domain of axin selectively interacts with Galpha12 but not Galpha13..
70:1461-1468.
2006
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Molecular determinants in the second intracellular loop of the 5-hydroxytryptamine-1A receptor for G-protein coupling..
69:1518-1526.
2006
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Erratum: TRPV1b, a functional human vanilloid receptor splice variant (Molecular Pharmacology (2004) 67 (1119-1127)).
67:1818.
2005
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Beta-arrestin 2-dependent angiotensin II type 1A receptor-mediated pathway of chemotaxis..
67:1229-1236.
2005
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TRPV1b, a functional human vanilloid receptor splice variant..
67:1119-1127.
2005
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Identification of amino acid residues in the insect sodium channel critical for pyrethroid binding..
67:513-522.
2005
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Reciprocal signaling between the transcriptional co-factor Eya2 and specific members of the Galphai family..
66:1325-1331.
2004
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Ligand-binding residues integrate affinity and efficacy in the NMDA receptor..
66:209-219.
2004
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Relative opioid efficacy is determined by the complements of the G protein-coupled receptor desensitization machinery..
66:106-112.
2004
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Subunit composition and pharmacology of two classes of striatal presynaptic nicotinic acetylcholine receptors mediating dopamine release in mice..
65:1526-1535.
2004
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The type 1 angiotensin II receptor tail affects receptor targeting, internalization, and membrane fusion properties..
65:362-369.
2004
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Center stage for the serotonin transporter: a gain-of-function polymorphism in persons with obsessive-compulsive disorder..
64:196-198.
2003
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Regulation of G protein-coupled receptor kinases and arrestins during receptor desensitization..
63:9-18.
2003
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Discovery of novel targets of quinoline drugs in the human purine binding proteome..
62:1364-1372.
2002
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Dancing with different partners: protein kinase a phosphorylation of seven membrane-spanning receptors regulates their G protein-coupling specificity..
62:971-974.
2002
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The Ca(2+) channel antagonists mibefradil and pimozide inhibit cell growth via different cytotoxic mechanisms..
62:210-219.
2002
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Vascular-targeted overexpression of G protein-coupled receptor kinase-2 in transgenic mice attenuates beta-adrenergic receptor signaling and increases resting blood pressure..
61:749-758.
2002
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Caspase-dependent cleavage of carbamoyl phosphate synthetase II during apoptosis..
61:569-577.
2002
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Transcriptional control of intestinal cytochrome P-4503A by 1alpha,25-dihydroxy vitamin D3..
60:1399-1406.
2001
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Reversal of physiological stress-induced resistance to topoisomerase II inhibitors using an inducible phosphorylation site-deficient mutant of I kappa B alpha..
60:559-567.
2001
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Fibronectin-mediated hepatocyte shape change reprograms cytochrome P450 2C11 gene expression via an integrin-signaled induction of ribonuclease activity..
58:976-981.
2000
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Interaction of methoxychlor and related compounds with estrogen receptor alpha and beta, and androgen receptor: structure-activity studies..
58:852-858.
2000
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5-Iodo-A-85380, an alpha4beta2 subtype-selective ligand for nicotinic acetylcholine receptors..
57:642-649.
2000
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Characterization of differences between rapid agonist-dependent phosphorylation and phorbol ester-mediated phosphorylation of human substance P receptor in intact cells..
55:855-862.
1999
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Constitutively active alpha-1b adrenergic receptor mutants display different phosphorylation and internalization features..
55:339-347.
1999
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Aspirin inhibits tumor necrosis factoralpha gene expression in murine tissue macrophages..
52:421-429.
1997
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Selective inhibition of adenylyl cyclase type V by the dopamine D3 receptor..
52:508-514.
1997
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Synergistic regulation of beta2-adrenergic receptor sequestration: intracellular complement of beta-adrenergic receptor kinase and beta-arrestin determine kinetics of internalization..
51:800-808.
1997
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Internal trafficking and surface mobility of a functionally intact beta2-adrenergic receptor-green fluorescent protein conjugate..
51:177-184.
1997
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The role of inactivation in open-channel block of the sodium channel: studies with inactivation-deficient mutant channels..
50:1643-1650.
1996
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Calcineurin mutants render T lymphocytes resistant to cyclosporin A..
50:506-511.
1996
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A novel nonopioid action of enkephalins: competitive inhibition of the mammalian brain high affinity L-proline transporter..
49:1033-1041.
1996
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Buthionine sulfoximine induction of gamma-L-glutamyl-L-cysteine synthetase gene expression, kinetics of glutathione depletion and resynthesis, and modulation of carmustine-induced DNA-DNA cross-linking and cytotoxicity in human glioma cells..
49:1012-1020.
1996
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5-Hydroxytryptamine2A receptors expressed in rat renal mesangial cells inhibit cyclic AMP accumulation..
48:230-237.
1995
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Agonist-dependent phosphorylation of the mouse delta-opioid receptor: involvement of G protein-coupled receptor kinases but not protein kinase C..
48:173-177.
1995
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N-methyl-D-aspartate receptors activate transcription of c-fos and NGFI-A by distinct phospholipase A2-requiring intracellular signaling pathways..
47:1119-1125.
1995
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Expression of alpha 1-adrenergic receptor subtype mRNA in rat tissues and human SK-N-MC neuronal cells: implications for alpha 1-adrenergic receptor subtype classification..
46:221-226.
1994
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High affinity agonist binding to the dopamine D3 receptor: chimeric receptors delineate a role for intracellular domains..
46:352-356.
1994
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Intranigral administration of D2 dopamine receptor antisense oligodeoxynucleotides establishes a role for nigrostriatal D2 autoreceptors in the motor actions of cocaine..
46:51-57.
1994
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Cloning of the human glycine transporter type 1: molecular and pharmacological characterization of novel isoform variants and chromosomal localization of the gene in the human and mouse genomes..
45:608-617.
1994
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Negative antagonists promote an inactive conformation of the beta 2-adrenergic receptor..
45:390-394.
1994
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Localization of mRNA for three distinct alpha 1-adrenergic receptor subtypes in human tissues: implications for human alpha-adrenergic physiology..
45:171-175.
1994
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Cloning and characterization of the opossum kidney cell D1 dopamine receptor: expression of identical D1A and D1B dopamine receptor mRNAs in opossum kidney and brain..
44:918-925.
1993
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Characterization of alpha 2-adrenergic receptor subtype-specific antibodies..
43:444-450.
1993
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8-hydroxy-2-(di-n-propylamino)tetralin-responsive 5-hydroxytryptamine4-like receptor expressed in bovine pulmonary artery smooth muscle cells..
42:817-825.
1992
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Cloning, pharmacological characterization, and chromosome assignment of the human dopamine transporter..
42:383-390.
1992
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Pharmacological characteristics of alpha 2-adrenergic receptors: comparison of pharmacologically defined subtypes with subtypes identified by molecular cloning..
42:1-5.
1992
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Functionally relevant gamma-aminobutyric acidA receptors: equivalence between receptor affinity (Kd) and potency (EC50)?.
41:1124-1129.
1992
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The alpha 1C-adrenergic receptor: characterization of signal transduction pathways and mammalian tissue heterogeneity..
40:619-626.
1991
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Patterns of internal and external tetraethylammonium block in four homologous K+ channels..
40:299-307.
1991
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5-Lipoxygenase-activating protein is the target of a quinoline class of leukotriene synthesis inhibitors..
40:22-27.
1991
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Effect of anti-human immunodeficiency virus nucleoside analogs on mitochondrial DNA and its implication for delayed toxicity..
39:625-628.
1991
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cAMP analogs inhibit gamma-aminobutyric acid-gated chloride flux and activate protein kinase A in brain synaptoneurosomes..
39:370-375.
1991
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Mutations of the human beta 2-adrenergic receptor that impair coupling to Gs interfere with receptor down-regulation but not sequestration..
39:192-198.
1991
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Regulation of responsiveness at D2 dopamine receptors by receptor desensitization and adenylyl cyclase sensitization..
39:55-63.
1991
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The α(1C)-adrenergic receptor: Characterization of signal transduction pathways and mammalian tissue heterogeneity.
40:619-626.
1991
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Expression of three alpha 2-adrenergic receptor subtypes in rat tissues: implications for alpha 2 receptor classification..
38:599-603.
1990
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Evidence that zinc inhibits N-methyl-D-aspartate receptor-gated ion channel activation by noncompetitive antagonism of glycine binding..
38:14-19.
1990
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Differential expression of gamma-aminobutyric acidA receptor subunits..
37:652-657.
1990
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Cytochrome P450IA1 induction and localization in endothelium of vertebrate (teleost) heart..
36:723-729.
1989
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Altered patterns of agonist-stimulated cAMP accumulation in cells expressing mutant beta 2-adrenergic receptors lacking phosphorylation sites..
36:641-646.
1989
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Glycine regulation of the N-methyl-D-aspartate receptor-gated ion channel in hippocampal membranes..
36:273-279.
1989
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Identification of the ligand-binding subunit of the human 5-hydroxytryptamine1A receptor with N-(p-azido-m-[125I] iodophenethyl)spiperone, a high affinity radioiodinated photoaffinity probe..
36:15-21.
1989
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The porcine heart M2 muscarinic receptor: agonist-induced phosphorylation and comparison of properties with the chick heart receptor..
35:553-558.
1989
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N-methyl-D-aspartate receptor regulation of uncompetitive antagonist binding in rat brain membranes: kinetic analysis..
34:250-255.
1988
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Isobutylmethylxanthine stimulates adenylate cyclase by blocking the inhibitory regulatory protein, Gi..
34:37-41.
1988
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Interaction of the antifolate antibiotic trimethoprim with phosphatidylcholine membranes: a 13C and 31P nuclear magnetic resonance study..
33:551-558.
1988
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The new cardiotonic agent sulmazole is an A1 adenosine receptor antagonist and functionally blocks the inhibitory regulator, Gi..
33:441-448.
1988
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Induction of rat cytochrome P-450 3 and its mRNA by 3,4,5,3',4',5'-hexachlorobiphenyl..
33:272-278.
1988
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Binding of [125I]-N-(p-aminophenethyl)spiroperidol to the D-2 dopamine receptor in the neurointermediate lobe of the rat pituitary gland: a thermodynamic study..
33:163-169.
1988
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Expression of a human cDNA encoding the beta 2-adrenergic receptor in Chinese hamster fibroblasts (CHW): functionality and regulation of the expressed receptors..
33:133-139.
1988
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Suppression of the constitutive, male-specific rat hepatic cytochrome P-450 2c and its mRNA by 3,4,5,3',4',5'-hexachlorobiphenyl and 3-methylcholanthrene..
32:340-347.
1987
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Identification of the binding subunit of the D1-dopamine receptor by photoaffinity crosslinking..
31:129-134.
1987
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γ-Aminobutyric acid (GABA)- and barbiturate-mediated 36
Cl-uptake in rat brain synaptoneurosomes: Evidence for rapid desensitization of the GABA receptor-coupled chloride ion channel.
30:419-426.
1986
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gamma-Aminobutyric acid (GABA)- and barbiturate-mediated 36Cl- uptake in rat brain synaptoneurosomes: evidence for rapid desensitization of the GABA receptor-coupled chloride ion channel..
30:419-426.
1986
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Characterization of DNA lesions induced by CaCrO4 in synchronous and asynchronous cultured mammalian cells..
29:606-613.
1986
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Phasic ion channel blockade. A kinetic model and parameter estimation procedure..
28:348-356.
1985
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Homologous desensitization of the beta-adrenergic receptor. Functional integrity of the desensitized receptor from mammalian lung..
28:237-245.
1985
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Covalent labeling of the beta-adrenergic ligand-binding site with para-(bromoacetamidyl)benzylcarazolol. A highly potent beta-adrenergic affinity label..
27:499-506.
1985
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Photoaffinity cross-linking of a radioiodinated probe, 125I-A55453, into alpha 1-adrenergic receptors..
26:187-195.
1984
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Barbiturate effects on acetylcholine-activated channels in Aplysia neurons..
24:449-457.
1983
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[3H]acetylcholine binding sites in brain. Effect of disulfide bond modification..
24:387-391.
1983
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Growth inhibition and metallothionein induction in cadmium-resistant cells by essential and non-essential metals..
24:77-83.
1983
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Regulation of insulin receptors in frog erythrocytes by insulin and concanavalin A. Evidence for discrete classes of insulin binding sites..
22:619-626.
1982
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Dopamine receptor of the porcine anterior pituitary gland. Effects of N-ethylmaleimide and heat on ligand binding mimic the effects of guanine nucleotides..
22:298-303.
1982
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Dopamine receptor of the porcine anterior pituitary gland. Evidence for two affinity states discriminated by both agonists and antagonists..
22:290-297.
1982
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Inhibition of microsomal oxidative drug metabolism by 1,4-bis (2-[(2-hydroxyethyl)amino]-ethylamino)-9,10-anthracenedione diacetate, a new antineoplastic agent..
22:471-478.
1982
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Nicotinic cholinergic receptors labeled by [3H]acetylcholine in rat brain..
22:56-62.
1982
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Validation and statistical analysis of a computer modeling method for quantitative analysis of radioligand binding data for mixtures of pharmacological receptor subtypes..
21:5-16.
1982
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Solubilization of a [3H]cimetidine binding site from rat brains. A clonidine-sensitive H-2 receptor subtype?.
20:240-243.
1981
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Determination of subtype selectivity of alpha-adrenergic antagonists: comparison of selective and nonselective radioligands..
20:28-34.
1981
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Alternative explanation for the apparent "two-step" binding kinetics of high-affinity racemic antagonist radioligands..
19:509-512.
1981
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Anomalous equilibrium binding properties of high-affinity racemic radioligands..
19:205-216.
1981
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Involvement of radical species in the oxidation of aminopyrine and 4-aminoantipyrine by cumene hydroperoxide in rat liver microsomes..
19:146-152.
1981
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Regulation of ornithine decarboxylase activity in the developing heart of euthyroid or hyperthyroid rats..
18:247-252.
1980
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Absence of metabolite formation during nitroglycerin-induced relaxation of isolated blood vessels..
18:112-116.
1980
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A quantitative analysis of beta-adrenergic receptor interactions: resolution of high and low affinity states of the receptor by computer modeling of ligand binding data..
17:14-23.
1980
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Multiple reactive sulfhydryl groups modulate the function of adenylate cyclase coupled beta-adrenergic receptors..
16:709-718.
1979
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Regulation of rat heart ornithine decarboxylase: change in affinity for ornithine evoked by neuronal, hormonal, and ontogenetic stimuli..
16:504-512.
1979
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Agonist-specific effects of guanine nucleotides on alpha-adrenergic receptors in human platelets..
16:61-68.
1979
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Interaction of halothane with lipid bilayers..
16:163-170.
1979
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Quantitative resolution of beta-adrenergic receptor subtypes by selective ligand binding: application of a computerized model fitting technique..
16:1-9.
1979
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Selective alteration in high affinity agonist binding: a mechanism of beta-adrenergic receptor desensitization..
16:10-20.
1979
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Structural characteristics for inhibition of [3H] norepinephrine uptake into rat brain synaptic vesicles by beta-carboline, indolealkylamine, phenethylamine and n-alkylamine derivatives..
15:607-619.
1979
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Ionic and nucleotide cofactor requirements for uptake of [3H]norepinephrine by rat brain synaptic vesicle preparations..
14:868-878.
1978
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Agonist-specific effects of monovalent and divalent cations on adenylate cyclase-coupled alpha adrenergic receptors in rabbit platelets..
14:540-548.
1978
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A desensitized state of the beta adrenergic receptor not associated with high-affinity agonist occupancy..
14:376-380.
1978
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Agonist-specific alterations in receptor binding affinity associated with solubilization of turkey erythrocyte membrane beta adrenergic receptors..
14:370-375.
1978
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Molecular pharmacology of alpha adrenergic receptors: utilization of [3H]dihydroergocryptine binding in the study of pharmacological receptor alterations..
13:304-313.
1977
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Regulation of beta adrenergic receptors in isolated frog erythrocyte plasma membranes..
13:291-303.
1977
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Adenylate cyclase-coupled beta adrenergic receptors effect of membrane lipid-perturbing agents on receptor binding and enzyme stimulation by catecholamines..
12:559-567.
1976
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X-ray crystal structure and conformation of a spin-labeled acetylcholine, DL-4-[N,N-dimethyl-n-(ethan-2'-olacetate)amino]-2,2,6,6-tetramethylpiperidine-1-oxyliodide..
12:590-597.
1976
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Regulation of adenylate cyclase-coupled beta adrenergic receptor binding sites by beta adrenergic catecholamines in vitro..
12:409-419.
1976
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Structure-activity relationships of adenylate cyclase-coupled beta adrenergic receptors: determination by direct binding studies..
12:16-31.
1976
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(3H)-Propranolol binding sites in myocardial membranes: nonidentity with beta adrenergic receptors..
10:450-456.
1974
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Reserpine-like effects of harmine on isolated adrenal medullary vesicles..
9:748-755.
1973
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Recovery of rat adrenal amine stores after insulin administration..
9:105-116.
1973
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Uptake, storage, and distribution of amines in bovine adrenal medullary vesicles..
7:581-592.
1971
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Compartmental analysis of amine storage in bovine adrenal medullary granules..
7:308-316.
1971