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Publication Venue For
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Design, synthesis, and antiviral activity of phenylalanine derivatives as HIV-1 capsid inhibitors..
48:116414.
2021
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Labeling a TCO-functionalized single domain antibody fragment with 18F via inverse electron demand Diels Alder cycloaddition using a fluoronicotinyl moiety-bearing tetrazine derivative..
28:115634.
2020
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Identification of potent pyrazole based APELIN receptor (APJ) agonists..
28:115237.
2020
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Identification of DK419, a potent inhibitor of Wnt/β-catenin signaling and colorectal cancer growth..
26:5435-5442.
2018
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Design, synthesis, and functional assessment of Cmpd-15 derivatives as negative allosteric modulators for the β2-adrenergic receptor..
26:2320-2330.
2018
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Fluorine-18 labeling of an anti-HER2 VHH using a residualizing prosthetic group via a strain-promoted click reaction: Chemistry and preliminary evaluation..
26:1939-1949.
2018
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Design, synthesis and biological evaluation of GPR55 agonists..
25:4355-4367.
2017
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Benzimidazole inhibitors from the Niclosamide chemotype inhibit Wnt/β-catenin signaling with selectivity over effects on ATP homeostasis..
25:1804-1816.
2017
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Structure-activity studies of Wnt/β-catenin inhibition in the Niclosamide chemotype: Identification of derivatives with improved drug exposure..
23:5829-5838.
2015
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4,4'-Unsymmetrically substituted 3,3'-biphenyl alpha helical proteomimetics as potential coactivator binding inhibitors..
22:917-926.
2014
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SIB-DOTA: a trifunctional prosthetic group potentially amenable for multi-modal labeling that enhances tumor uptake of internalizing monoclonal antibodies..
20:6929-6939.
2012
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Identification of a novel Smoothened antagonist that potently suppresses Hedgehog signaling..
20:6751-6757.
2012
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Covalent protein-oligonucleotide conjugates by copper-free click reaction..
20:4532-4539.
2012
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A highly selective Hsp90 affinity chromatography resin with a cleavable linker..
20:3298-3305.
2012
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Syntheses, structures and antibiotic activities of LpxC inhibitors based on the diacetylene scaffold..
19:852-860.
2011
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Anti-AIDS agents 79. Design, synthesis, molecular modeling and structure-activity relationships of novel dicamphanoyl-2',2'-dimethyldihydropyranochromone (DCP) analogs as potent anti-HIV agents..
18:6678-6689.
2010
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Conjugates of betulin derivatives with AZT as potent anti-HIV agents..
18:6451-6469.
2010
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Anti-AIDS agents 82: synthesis of seco-(3'R,4'R)-3',4'-di-O-(S)-camphanoyl-(+)-cis-khellactone (DCK) derivatives as novel anti-HIV agents..
18:4363-4373.
2010
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Psammaplin A as a general activator of cell-based signaling assays via HDAC inhibition and studies on some bromotyrosine derivatives..
17:2189-2198.
2009
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Tyrosine-sulfate isosteres of CCR5 N-terminus as tools for studying HIV-1 entry..
16:10113-10120.
2008
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Synthesis and proteasome inhibition of glycyrrhetinic acid derivatives..
16:6696-6701.
2008
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Synthesis, fluorine-18 radiolabeling, and in vitro characterization of 1-iodophenyl-N-methyl-N-fluoroalkyl-3-isoquinoline carboxamide derivatives as potential PET radioligands for imaging peripheral benzodiazepine receptor..
16:6145-6155.
2008