Spiperone
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Subject Areas on Research
- 3-(2'-[18F]fluoroethyl)spiperone, a potent dopamine antagonist: synthesis, structural analysis and in-vivo utilization in humans.
- A novel radioiodinated high affinity ligand for the D2-dopamine receptor. Characterization of its binding in bovine anterior pituitary membranes.
- Affinity chromatography of the anterior pituitary D2-dopamine receptor.
- Agonist binding promotes a guanine nucleotide reversible increase in the apparent size of the bovine anterior pituitary dopamine receptors.
- Binding of [125I]-N-(p-aminophenethyl)spiroperidol to the D-2 dopamine receptor in the neurointermediate lobe of the rat pituitary gland: a thermodynamic study.
- Chlorpromazine methiodide-induced barrel rotation: an antimuscarinic effect.
- Chronic lithium administration has no effect on haloperidol-induced supersensitivity of pre- and postsynaptic dopamine receptors in rat brain.
- Chronic sulpiride increased 3H-spiperone binding and calmodulin dependent phosphorylation in rat striatum.
- Clonazepam-induced up-regulation of serotonin1 and serotonin2 binding sites in rat frontal cortex.
- Colchicine administered into the area of the nucleus basalis decreases cortical nicotinic cholinergic receptors labelled by [3H]-acetylcholine.
- Comparative antidopaminergic properties of thioridazine, mesoridazine and sulforidazine on the corpus striatum.
- D2 dopamine receptors in the human retina: cloning of cDNA and localization of mRNA.
- Direct radioligand measurement of dopamine receptors in the anterior pituitary gland.
- Dopamine receptor of the porcine anterior pituitary gland. Effects of N-ethylmaleimide and heat on ligand binding mimic the effects of guanine nucleotides.
- Dopamine receptor of the porcine anterior pituitary gland. Evidence for two affinity states discriminated by both agonists and antagonists.
- Dopamine receptor of the porcine anterior pituitary gland. Solubilization and characterization.
- Dopamine receptors status after unilateral nigral 6-OHDA lesion. Autoradiographic and in situ hybridization study in the rat brain.
- Effects of intrastriatal infusion of D2 and D3 dopamine receptor preferring antagonists on dopamine release in rat dorsal striatum (in vivo microdialysis study).
- Electroconvulsive treatment and haloperidol: effects on pre- and postsynaptic dopamine receptors in rat brain.
- Guanine nucleotides regulate both dopaminergic agonist and antagonist binding in porcine anterior pituitary.
- Identification of the D2-dopamine receptor binding subunit in several mammalian tissues and species by photoaffinity labeling.
- Identification of the ligand-binding subunit of the human 5-hydroxytryptamine1A receptor with N-(p-azido-m-[125I] iodophenethyl)spiperone, a high affinity radioiodinated photoaffinity probe.
- Lack of potency of metoclopramide's metabolites in various dopaminergic models.
- Neurotensin interacts with dopaminergic neurons in rat brain.
- No-carrier-added 3-(2'-[18F]fluoroethyl)spiperone, a new dopamine receptor-binding tracer for positron emission tomography.
- Pharmacologic evaluation of dopaminergic receptor blockade by metoclopramide.
- Photoaffinity labeling of the D2-dopamine receptor using a novel high affinity radioiodinated probe.
- Purification and characterization of the D2-dopamine receptor from bovine anterior pituitary.
- Reserpine-induced up-regulation of dopamine D2 receptors in the rat striatum is enhanced by denervation but not by chronic receptor blockade.
- Solubilization and characterization of D2-dopamine receptors in an estrone-induced, prolactin-secreting rat pituitary adenoma.
- Studies of dopamine pharmacology in molluscs.
- The effect of chronic L-dopa administration on supersensitive pre- and postsynaptic dopaminergic receptors in rat brain.
- The effects of chronic bromocriptine treatment on behaviour and dopamine receptor binding in the rat striatum.