Receptors, Neurotensin
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Subject Areas on Research
- Discovery of β-Arrestin Biased, Orally Bioavailable, and CNS Penetrant Neurotensin Receptor 1 (NTR1) Allosteric Modulators.
- Identification and functional characterization of a stable, centrally active derivative of the neurotensin (8-13) fragment as a potential first-in-class analgesic.
- Imidazole-derived agonists for the neurotensin 1 receptor.
- ML314: A Biased Neurotensin Receptor Ligand for Methamphetamine Abuse.
- Molecular determinants underlying the formation of stable intracellular G protein-coupled receptor-beta-arrestin complexes after receptor endocytosis*.
- Neurotensin Receptor Allosterism Revealed in Complex with a Biased Allosteric Modulator.
- Neurotensin receptor 1-biased ligand attenuates neurotensin-mediated excitation of ventral tegmental area dopamine neurons and dopamine release in the nucleus accumbens.
- Triphenylmethane dye activation of beta-arrestin.
- β-Arrestin-Biased Allosteric Modulator of NTSR1 Selectively Attenuates Addictive Behaviors.