Non-peptidic, non-prenylic inhibitors of the prenyl protein-specific protease Rce1.
Publication
, Journal Article
Schlitzer, M; Winter-Vann, A; Casey, PJ
Published in: Bioorg Med Chem Lett
February 12, 2001
Several compounds designed as bisubstrate analogues of protein farnesyltransferase inhibited the prenyl protein-specific protease Rce1, qualifying them as lead structures for a novel class of non-peptidic, non-prenylic inhibitors of this protease.
Duke Scholars
Published In
Bioorg Med Chem Lett
DOI
ISSN
0960-894X
Publication Date
February 12, 2001
Volume
11
Issue
3
Start / End Page
425 / 427
Location
England
Related Subject Headings
- Structure-Activity Relationship
- Protease Inhibitors
- Peptides
- Molecular Mimicry
- Medicinal & Biomolecular Chemistry
- Inhibitory Concentration 50
- Humans
- Farnesyltranstransferase
- Endopeptidases
- Combinatorial Chemistry Techniques
Citation
APA
Chicago
ICMJE
MLA
NLM
Schlitzer, M., Winter-Vann, A., & Casey, P. J. (2001). Non-peptidic, non-prenylic inhibitors of the prenyl protein-specific protease Rce1. Bioorg Med Chem Lett, 11(3), 425–427. https://doi.org/10.1016/s0960-894x(00)00685-5
Schlitzer, M., A. Winter-Vann, and P. J. Casey. “Non-peptidic, non-prenylic inhibitors of the prenyl protein-specific protease Rce1.” Bioorg Med Chem Lett 11, no. 3 (February 12, 2001): 425–27. https://doi.org/10.1016/s0960-894x(00)00685-5.
Schlitzer M, Winter-Vann A, Casey PJ. Non-peptidic, non-prenylic inhibitors of the prenyl protein-specific protease Rce1. Bioorg Med Chem Lett. 2001 Feb 12;11(3):425–7.
Schlitzer, M., et al. “Non-peptidic, non-prenylic inhibitors of the prenyl protein-specific protease Rce1.” Bioorg Med Chem Lett, vol. 11, no. 3, Feb. 2001, pp. 425–27. Pubmed, doi:10.1016/s0960-894x(00)00685-5.
Schlitzer M, Winter-Vann A, Casey PJ. Non-peptidic, non-prenylic inhibitors of the prenyl protein-specific protease Rce1. Bioorg Med Chem Lett. 2001 Feb 12;11(3):425–427.
Published In
Bioorg Med Chem Lett
DOI
ISSN
0960-894X
Publication Date
February 12, 2001
Volume
11
Issue
3
Start / End Page
425 / 427
Location
England
Related Subject Headings
- Structure-Activity Relationship
- Protease Inhibitors
- Peptides
- Molecular Mimicry
- Medicinal & Biomolecular Chemistry
- Inhibitory Concentration 50
- Humans
- Farnesyltranstransferase
- Endopeptidases
- Combinatorial Chemistry Techniques