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Structure-guided design and synthesis of C22- and C32-modified FK520 analogs with enhanced activity against human pathogenic fungi.

Publication ,  Preprint
Dome, PA; Jeong, P; Nam, G; Jang, H; Rivera, A; Averette, AF; Park, E; Liao, T-C; Ciofani, M; Wu, J; Chi, J-TA; Venters, RA; Park, H-J ...
November 8, 2024

Duke Scholars

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November 8, 2024
 

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Dome, P. A., Jeong, P., Nam, G., Jang, H., Rivera, A., Averette, A. F., … Hong, J. (2024). Structure-guided design and synthesis of C22- and C32-modified FK520 analogs with enhanced activity against human pathogenic fungi. https://doi.org/10.1101/2024.09.27.615491
Dome, Patrick A., Pyeonghwa Jeong, Gibeom Nam, Hongjun Jang, Angela Rivera, Anna Floyd Averette, Eunchong Park, et al. “Structure-guided design and synthesis of C22- and C32-modified FK520 analogs with enhanced activity against human pathogenic fungi.,” November 8, 2024. https://doi.org/10.1101/2024.09.27.615491.
Dome PA, Jeong P, Nam G, Jang H, Rivera A, Averette AF, Park E, Liao T-C, Ciofani M, Wu J, Chi J-TA, Venters RA, Park H-J, Steinbach WJ, Juvvadi PR, Heitman J, Hong J. Structure-guided design and synthesis of C22- and C32-modified FK520 analogs with enhanced activity against human pathogenic fungi. 2024.

DOI

Publication Date

November 8, 2024