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A randomized comparative study to determine the effect of omeprazole on the peak serum concentration of itraconazole oral solution.

Publication ,  Journal Article
Johnson, MD; Hamilton, CD; Drew, RH; Sanders, LL; Pennick, GJ; Perfect, JR
Published in: J Antimicrob Chemother
February 2003

To determine the effect of omeprazole on peak serum concentrations (C(max)) of itraconazole oral solution (IOS), we carried out a randomized, open-label, prospective, crossover study. Fifteen healthy, non-pregnant adults received a single dose of IOS 400 mg on two occasions, at least 7 days apart, with omeprazole 40 mg nightly for 7 days before either IOS dose 1 or 2. C(max), time to C(max) (T(max)) and AUC(0-8) were determined for itraconazole and its active metabolite, hydroxyitraconazole, for each dose and compared. Omeprazole did not significantly affect the C(max), T(max) or AUC(0-8) of itraconazole or hydroxyitraconazole when administered as IOS.

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Published In

J Antimicrob Chemother

DOI

ISSN

0305-7453

Publication Date

February 2003

Volume

51

Issue

2

Start / End Page

453 / 457

Location

England

Related Subject Headings

  • Pharmaceutical Solutions
  • Omeprazole
  • Middle Aged
  • Microbiology
  • Male
  • Itraconazole
  • Humans
  • Female
  • Drug Interactions
  • Biotransformation
 

Citation

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Johnson, M. D., Hamilton, C. D., Drew, R. H., Sanders, L. L., Pennick, G. J., & Perfect, J. R. (2003). A randomized comparative study to determine the effect of omeprazole on the peak serum concentration of itraconazole oral solution. J Antimicrob Chemother, 51(2), 453–457. https://doi.org/10.1093/jac/dkg089
Johnson, Melissa D., Carol D. Hamilton, Richard H. Drew, Linda L. Sanders, Gennethel J. Pennick, and John R. Perfect. “A randomized comparative study to determine the effect of omeprazole on the peak serum concentration of itraconazole oral solution.J Antimicrob Chemother 51, no. 2 (February 2003): 453–57. https://doi.org/10.1093/jac/dkg089.
Johnson MD, Hamilton CD, Drew RH, Sanders LL, Pennick GJ, Perfect JR. A randomized comparative study to determine the effect of omeprazole on the peak serum concentration of itraconazole oral solution. J Antimicrob Chemother. 2003 Feb;51(2):453–7.
Johnson, Melissa D., et al. “A randomized comparative study to determine the effect of omeprazole on the peak serum concentration of itraconazole oral solution.J Antimicrob Chemother, vol. 51, no. 2, Feb. 2003, pp. 453–57. Pubmed, doi:10.1093/jac/dkg089.
Johnson MD, Hamilton CD, Drew RH, Sanders LL, Pennick GJ, Perfect JR. A randomized comparative study to determine the effect of omeprazole on the peak serum concentration of itraconazole oral solution. J Antimicrob Chemother. 2003 Feb;51(2):453–457.
Journal cover image

Published In

J Antimicrob Chemother

DOI

ISSN

0305-7453

Publication Date

February 2003

Volume

51

Issue

2

Start / End Page

453 / 457

Location

England

Related Subject Headings

  • Pharmaceutical Solutions
  • Omeprazole
  • Middle Aged
  • Microbiology
  • Male
  • Itraconazole
  • Humans
  • Female
  • Drug Interactions
  • Biotransformation